DSA
Kilo KaybıKapsamlı Çalışılmış3 çalışma

Cagrilintide

Long-Acting Amylin Receptor Agonist | Weight Loss & Diabetes

Novel long-acting lipidated amylin analog functioning as dual amylin and calcitonin receptor agonist for weight management and type 2 diabetes. Phase 3 trials demonstrate 22.7% weight loss with CagriSema combination.

Yarı ömür
~7 days (159-195 hours)
Sıklık
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Döngü
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Doz
2.4mg weekly (after escalation)
Cagrilintide 2D chemical structure

M.W.: 4,409.01 Da

PubChem 2D yapı diyagramı

DEEP ARCHIVESUPPLEMENTCagrilintideLong-Acting Amylin Recepto…PURITY: 99% HPLCRUO: Research Use OnlyREF CAG-431-DSAM.W. 4,409.01 DaNOT FOR HUMAN OR VETERINARY USE

Referans illüstrasyonu — ürün listesi değildir

Etki Mekanizması

Subcutaneous injection enables optimal bioavailability, targeting dual amylin and calcitonin receptors for satiety and metabolic regulation. Enhances insulin sensitivity and controls gastric emptying.

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Novel long-acting lipidated amylin analog functioning as dual amylin and calcitonin receptor agonist for weight management and type 2 diabetes. Phase 3 trials demonstrate 22.7% weight loss with CagriSema combination.

Moleküler Veri

Tür
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Moleküler ağırlık
4,409.01 Da

1000 mcg = 1 mg

1 = her gün · 7 = haftalık

Süre (gün)

Araştırma Endikasyonları

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effective

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most effective

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most effective

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most effective

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effective

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effective

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Doz Protokolleri

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HedefDozSıklıkYol
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Etkileşimler

++
Semaglutide
synergistic

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+
Tirzepatide
compatible

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Retatrutide
monitor

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Metformin
compatible

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SGLT2 Inhibitors
compatible

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+
Pramlintide
compatible

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Oral Contraceptives
monitor

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Ne Beklenmeli

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