Tirzepatide
Dual GIP/GLP-1 Receptor Agonist | Weight Loss & Diabetes
Revolutionary dual receptor agonist FDA-approved for type 2 diabetes and chronic weight management. Demonstrates efficacy superior to single-mechanism alternatives with 15-22% body weight reduction in clinical trials. The first-in-class dual GIP/GLP-1 agonist provides enhanced metabolic benefits compared to GLP-1-only medications.
Moleküler Gösterim
M.W.: 4,813.55 Da
PubChem 2D yapı diyagramı
Referans Flakon
Referans illüstrasyonu — ürün listesi değildir
Etki Mekanizması
Dual agonist targeting both GIP and GLP-1 receptors, producing glucose-dependent insulin stimulation, delayed gastric emptying, glucagon suppression, and central satiety signaling via hypothalamic pathways.
Revolutionary dual receptor agonist FDA-approved for type 2 diabetes and chronic weight management. Demonstrates efficacy superior to single-mechanism alternatives with 15-22% body weight reduction in clinical trials. The first-in-class dual GIP/GLP-1 agonist provides enhanced metabolic benefits compared to GLP-1-only medications.
Moleküler Veri
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Doz Protokolleri
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| Hedef | Doz | Sıklık | Yol |
|---|---|---|---|
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Etkileşimler
Semaglutide
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Liraglutide
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Insulin
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Metformin
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CJC-1295
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Ipamorelin
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BPC-157
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5-Amino-1MQ
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Ne Beklenmeli
Yan Etkiler & Güvenlik
Yaygın Yan Etkiler
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Sık Sorulan Sorular
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Kaynaklar
- Tirzepatide Once Weekly for the Treatment of Obesity (SURMOUNT-1) — Jastreboff, A.M., et al.
- Tirzepatide versus Semaglutide Once Weekly in Patients with Type 2 Diabetes (SURPASS-2) — Frías, J.P., et al.
- Tirzepatide once weekly for the treatment of obesity in people with type 2 diabetes (SURMOUNT-2) — Garvey, W.T., et al.
- Cardiovascular Outcomes with Tirzepatide versus Dulaglutide in Type 2 Diabetes (SURPASS-CVOT) — Nicholls, S.J., et al.
- Tirzepatide for Obesity Treatment and Diabetes Prevention (SURMOUNT-1 3-Year Extension) — Jastreboff, A.M., et al.
- Tirzepatide for Heart Failure with Preserved Ejection Fraction and Obesity (SUMMIT) — Packer, M., et al.
- Tirzepatide as Compared with Semaglutide for the Treatment of Obesity (SURMOUNT-5) — Aronne, L.J., et al.
- Tirzepatide for the Treatment of Obstructive Sleep Apnea and Obesity (SURMOUNT-OSA) — Malhotra, A., et al.