DSA
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Hexarelin

Examorelin | Synthetic Growth Hormone Secretagogue

Hexarelin is one of the most potent synthetic growth hormone secretagogues available. It stimulates GH release by binding to the GHS-R1a receptor in the pituitary and hypothalamus, mimicking the action of ghrelin. Notably, Hexarelin demonstrates synergistic effects when combined with GHRH, producing GH responses greater than the arithmetic sum of either peptide alone. It also shows unique cardioprotective properties mediated through the CD36 receptor.

Yarı ömür
1-2 hours
Sıklık
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Döngü
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Doz
100-200 mcg per injection
Hexarelin 2D chemical structure

M.W.: 887 Da

PubChem 2D yapı diyagramı

DEEP ARCHIVESUPPLEMENTHexarelinExamorelin | Synthetic Gro…PURITY: 99% HPLCRUO: Research Use OnlyREF HEX-128-DSAM.W. 887 DaNOT FOR HUMAN OR VETERINARY USE

Referans illüstrasyonu — ürün listesi değildir

Etki Mekanizması

Hexarelin binds to the growth hormone secretagogue receptor 1a (GHS-R1a) in the brain and pituitary gland. This binding initiates a signaling cascade that stimulates somatotroph cells in the anterior pituitary to produce and release growth hormone. Hexarelin also has slight, dose-dependent effects on prolactin, ACTH, and cortisol release. Its cardioprotective effects are mediated through CD36 receptor activation and modulation of calcium channels in cardiomyocytes.

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Hexarelin is one of the most potent synthetic growth hormone secretagogues available. It stimulates GH release by binding to the GHS-R1a receptor in the pituitary and hypothalamus, mimicking the action of ghrelin. Notably, Hexarelin demonstrates synergistic effects when combined with GHRH, producing GH responses greater than the arithmetic sum of either peptide alone. It also shows unique cardioprotective properties mediated through the CD36 receptor.

Moleküler Veri

Tür
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Moleküler ağırlık
887 Da

1000 mcg = 1 mg

1 = her gün · 7 = haftalık

Süre (gün)

Araştırma Endikasyonları

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most effective

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most effective

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effective

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effective

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moderate

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moderate

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effective

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effective

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Doz Protokolleri

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HedefDozSıklıkYol
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Etkileşimler

++
CJC-1295
synergistic

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++
GHRH 1-29
synergistic

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+
GHRP-2
compatible

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+
GHRP-6
compatible

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+
Ipamorelin
compatible

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Ne Beklenmeli

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Yan Etkiler & Güvenlik

Yaygın Yan Etkiler

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