DSA
Kilo KaybıKapsamlı Çalışılmış3 çalışma

Survodutide

Dual GLP-1/Glucagon Receptor Agonist | Weight Loss & Diabetes

Investigational dual receptor agonist targeting metabolic disease through balanced GLP-1R and GCGR activation. Phase 2/3 clinical trials demonstrate superior weight loss and MASH treatment efficacy.

Yarı ömür
Approximately 6 days (109-115 hours)
Sıklık
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Döngü
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Doz
0.6mg starting, titrate up to 3.6-6.0mg weekly
Survodutide 2D chemical structure

M.W.: ~4,500 Da

PubChem 2D yapı diyagramı

DEEP ARCHIVESUPPLEMENTSurvodutideDual GLP-1/Glucagon Recept…PURITY: 99% HPLCRUO: Research Use OnlyREF SUR-382-DSAM.W. ~4,500 DaNOT FOR HUMAN OR VETERINARY USE

Referans illüstrasyonu — ürün listesi değildir

Etki Mekanizması

Dual agonism: GLP-1R reduces appetite and slows gastric emptying; GCGR increases energy expenditure and hepatic fat oxidation. EC50 0.52nM GCGR, 0.33nM GLP-1R.

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Investigational dual receptor agonist targeting metabolic disease through balanced GLP-1R and GCGR activation. Phase 2/3 clinical trials demonstrate superior weight loss and MASH treatment efficacy.

Moleküler Veri

Tür
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Moleküler ağırlık
~4,500 Da

1000 mcg = 1 mg

1 = her gün · 7 = haftalık

Süre (gün)

Araştırma Endikasyonları

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most effective

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most effective

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most effective

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most effective

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most effective

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effective

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Doz Protokolleri

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HedefDozSıklıkYol
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Etkileşimler

~
Semaglutide/Tirzepatide
monitor

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+
Metformin
compatible

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+
SGLT2 Inhibitors
compatible

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Sulfonylureas
monitor

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Insulin
monitor

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Oral Contraceptives
monitor

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+
Other Glucagon Agonists
compatible

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Ne Beklenmeli

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Yan Etkiler & Güvenlik

Yaygın Yan Etkiler

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Kaynaklar