Melanotan II
Synthetic Melanocortin Peptide | Tanning & Sexual Function
Melanotan II is a synthetic analog of alpha-melanocyte-stimulating hormone (α-MSH) that activates melanocortin receptors throughout the body. MC1R activation triggers melanin production for tanning, while MC4R affects sexual arousal and appetite control.
Moleküler Gösterim
PubChem 2D yapı diyagramı
Referans Flakon
Referans illüstrasyonu — ürün listesi değildir
Etki Mekanizması
Binds to melanocortin receptors (MC1R for tanning, MC4R for sexual function and appetite) to stimulate melanin production, enhance libido, and suppress appetite through hypothalamic pathways.
Melanotan II is a synthetic analog of alpha-melanocyte-stimulating hormone (α-MSH) that activates melanocortin receptors throughout the body. MC1R activation triggers melanin production for tanning, while MC4R affects sexual arousal and appetite control.
Moleküler Veri
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| Hedef | Doz | Sıklık | Yol |
|---|---|---|---|
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Kaynaklar
- Melanocortin Receptor Agonists, Penile Erection, and Sexual Motivation: Human Studies with Melanotan II — Wessells H, Levine N, Hadley ME, Dorr RT, Hruby VJ
- Increased Eumelanin Expression and Tanning Is Induced by a Superpotent Melanotropin [Nle4-D-Phe7]-alpha-MSH in Humans — Dorr RT, Lines R, Levine N, et al.
- Discovery that a Melanocortin Regulates Sexual Functions in Male and Female Humans — Hadley ME, Dorr RT
- Evaluation of Melanotan-II, a Superpotent Cyclic Melanotropic Peptide in a Pilot Phase-I Clinical Study — Dorr RT, Lines R, Levine N, Brooks C, et al.