DSA
Cilt & SaçFDA Onaylı3 çalışma

Melanotan I

Melanocortin Receptor Agonist

Synthetic analog of α-MSH that selectively targets MC1 receptors for melanin stimulation. FDA-approved as SCENESSE implant for erythropoietic protoporphyria (EPP). Research-grade injectable form enables flexible dosing versus the implant version.

Yarı ömür
~30 minutes
Sıklık
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Döngü
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Doz
Loading: 0.25-0.5mg daily; Maintenance: 0.25-0.5mg 2-3x weekly
Melanotan I 2D chemical structure

M.W.: 1646.88 Da

PubChem 2D yapı diyagramı

DEEP ARCHIVESUPPLEMENTMelanotan IMelanocortin Receptor Agon…PURITY: 99% HPLCRUO: Research Use OnlyREF MEL-232-DSAM.W. 1646.88 DaNOT FOR HUMAN OR VETERINARY USE

Referans illüstrasyonu — ürün listesi değildir

Etki Mekanizması

Subcutaneous injection delivers peptide directly into systemic circulation. Selectively activates MC1R receptors to stimulate melanin production. Short half-life of approximately 30 minutes necessitates multiple daily dosing for sustained effect.

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Synthetic analog of α-MSH that selectively targets MC1 receptors for melanin stimulation. FDA-approved as SCENESSE implant for erythropoietic protoporphyria (EPP). Research-grade injectable form enables flexible dosing versus the implant version.

Moleküler Veri

Tür
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Moleküler ağırlık
1646.88 Da

1000 mcg = 1 mg

1 = her gün · 7 = haftalık

Süre (gün)

Araştırma Endikasyonları

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most effective

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most effective

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effective

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most effective

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Doz Protokolleri

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HedefDozSıklıkYol
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Etkileşimler

+
Melanotan II
compatible

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++
UV Exposure
synergistic

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+
Beta-Carotene
compatible

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~
Tretinoin/Retinoids
monitor

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~
Photosensitizing Medications
monitor

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Ne Beklenmeli

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Yan Etkiler & Güvenlik

Yaygın Yan Etkiler

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Durdurma Belirtileri

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Kontrendikasyonlar

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    Kaynaklar