Semaglutide
GLP-1 Receptor Agonist | Weight Loss & Diabetes
Long-acting GLP-1 receptor agonist approved for type 2 diabetes and chronic weight management. Over 17,000 trial participants have demonstrated significant efficacy through appetite suppression and glycemic control. The 7-day half-life enables convenient weekly dosing.
Moleküler Gösterim
M.W.: 4,113.64 Da
PubChem 2D yapı diyagramı
Referans Flakon
Referans illüstrasyonu — ürün listesi değildir
Etki Mekanizması
Mimics native GLP-1, binding to receptors to stimulate glucose-dependent insulin secretion, suppress glucagon, slow gastric emptying, and reduce appetite via hypothalamic pathways.
Long-acting GLP-1 receptor agonist approved for type 2 diabetes and chronic weight management. Over 17,000 trial participants have demonstrated significant efficacy through appetite suppression and glycemic control. The 7-day half-life enables convenient weekly dosing.
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Kaynaklar
- Once-Weekly Semaglutide in Adults with Overweight or Obesity (STEP 1) — Wilding, J.P.H., et al.
- Semaglutide and Cardiovascular Outcomes in Obesity without Diabetes (SELECT) — Lincoff, A.M., et al.
- Semaglutide and Cardiovascular Outcomes in Patients with Type 2 Diabetes (SUSTAIN-6) — Marso, S.P., et al.
- Two-year effects of semaglutide in adults with overweight or obesity (STEP 5) — Garvey, W.T., et al.
- Oral Semaglutide and Cardiovascular Outcomes in Patients with Type 2 Diabetes (PIONEER 6) — Husain, M., et al.
- Once-Weekly Semaglutide in Adolescents with Obesity (STEP TEENS) — Weghuber, D., et al.
- Semaglutide in Patients with Heart Failure with Preserved Ejection Fraction and Obesity (STEP-HFpEF) — Kosiborod, M.N., et al.
- Effects of Semaglutide on Chronic Kidney Disease in Patients with Type 2 Diabetes (FLOW) — Perkovic, V., et al.
- Phase 3 Trial of Semaglutide in Metabolic Dysfunction-Associated Steatohepatitis (ESSENCE) — Sanyal, A.J., et al.