IGF-1 LR3
Modified Growth Factor Analog | Muscle Growth
IGF-1 LR3 is a synthetic 83-amino acid analog of insulin-like growth factor-1 that has never been approved for human use. The N-terminal extension and R3 substitution reduce binding protein interaction, maintaining elevated free circulating levels with ~3x greater potency than native IGF-1.
Moleküler Gösterim
PubChem 2D yapı diyagramı
Referans Flakon
Referans illüstrasyonu — ürün listesi değildir
Etki Mekanizması
Functions as a full IGF-1 receptor agonist activating PI3K/Akt/mTOR and MAPK/ERK pathways. The modifications prevent protein sequestration, maintaining elevated free circulating levels for extended anabolic effects.
IGF-1 LR3 is a synthetic 83-amino acid analog of insulin-like growth factor-1 that has never been approved for human use. The N-terminal extension and R3 substitution reduce binding protein interaction, maintaining elevated free circulating levels with ~3x greater potency than native IGF-1.
Moleküler Veri
Araştırma Endikasyonları
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Doz Protokolleri
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| Hedef | Doz | Sıklık | Yol |
|---|---|---|---|
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| MYMEMORY WARNING: YOU USED ALL AVAILABLE FREE TRANSLATIONS FOR TODAY. NEXT AVAILABLE IN 10 HOURS 45 MINUTES 46 SECONDS VISIT HTTPS://MYMEMORY.TRANSLATED.NET/DOC/USAGELIMITS.PHP TO TRANSLATE MORE | 40-60mcg | MYMEMORY WARNING: YOU USED ALL AVAILABLE FREE TRANSLATIONS FOR TODAY. NEXT AVAILABLE IN 11 HOURS 04 MINUTES 45 SECONDS VISIT HTTPS://MYMEMORY.TRANSLATED.NET/DOC/USAGELIMITS.PHP TO TRANSLATE MORE | MYMEMORY WARNING: YOU USED ALL AVAILABLE FREE TRANSLATIONS FOR TODAY. NEXT AVAILABLE IN 10 HOURS 47 MINUTES 25 SECONDS VISIT HTTPS://MYMEMORY.TRANSLATED.NET/DOC/USAGELIMITS.PHP TO TRANSLATE MORE |
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Etkileşimler
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Anabolic Steroids
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Kaynaklar
- Insulin-like growth factor-I (IGF-I) and especially IGF-I variants are anabolic in dexamethasone-treated rats — Tomas FM, Knowles SE, Owens PC, Chandler CS, Francis GL, Read LC, Ballard FJ
- Attenuated glucose-stimulated insulin secretion during an acute IGF-1 LR3 infusion into fetal sheep does not persist in isolated islets — Stremming J, White A, Galan HL, Brown LD
- Insulin-like growth factor I preserves host lean tissue mass in cancer cachexia — Ng EH, Rock CS, Lazarus DD, Stiaino-Coico L, Moldawer LL, Bhatt GR
- Circulating Insulin-like Growth Factor-I Concentrations and Risk of 30 Cancers: Prospective Analyses in UK Biobank — Murphy N, Knuppel A, Papadimitriou N, Martin RM, Tsilidis KK, Brennan P et al.