Dihexa
Synaptogenic Peptide | Cognitive Enhancement
Dihexa is a synthetic oligopeptide derived from angiotensin IV that potently enhances cognitive function by promoting synaptogenesis. It is 10 million times more potent than BDNF at promoting synapse formation through HGF/c-Met receptor activation.
Moleküler Gösterim
M.W.: 504.7 Da
PubChem 2D yapı diyagramı
Referans Flakon
Referans illüstrasyonu — ürün listesi değildir
Etki Mekanizması
Binds to hepatocyte growth factor (HGF) with high affinity (Kd = 65 pM) and potentiates its activity at c-Met receptor, activating PI3K/AKT pathways and promoting new synaptic connections with extraordinary potency.
Dihexa is a synthetic oligopeptide derived from angiotensin IV that potently enhances cognitive function by promoting synaptogenesis. It is 10 million times more potent than BDNF at promoting synapse formation through HGF/c-Met receptor activation.
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Kaynaklar
- Evaluation of Metabolically Stabilized Angiotensin IV Analogs as Procognitive/Antidementia Agents — McCoy AT, Benoist CC, Wright JW, Harding JW
- AngIV-Analog Dihexa Rescues Cognitive Impairment and Recovers Memory in the APP/PS1 Mouse via the PI3K/AKT Signaling Pathway — Gao Y, Zhang Y, Wang Z, et al.
- The Procognitive and Synaptogenic Effects of Angiotensin IV-Derived Peptides Are Dependent on Activation of the Hepatocyte Growth Factor/c-Met System — Benoist CC, Kawas LH, Zhu M, Bhatt D, Wright JW, Harding JW
- The Development of Small Molecule Angiotensin IV Analogs to Treat Alzheimer's and Parkinson's Diseases — Wright JW, Harding JW