MK-677
Ghrelin Receptor Agonist | Oral Growth Hormone Secretagogue
Oral compound activating ghrelin receptors to trigger growth hormone release while preserving natural production. Achieves superior oral bioavailability exceeding 60% with a 24-hour half-life, making it unique among GH secretagogues for its convenient once-daily oral dosing.
Moleküler Gösterim
M.W.: 624.77 Da
PubChem 2D yapı diyagramı
Referans Flakon
Referans illüstrasyonu — ürün listesi değildir
Etki Mekanizması
Selectively binds GHS-R1a receptors in hypothalamus and pituitary, triggering pulsatile growth hormone release while maintaining natural circadian patterns.
Oral compound activating ghrelin receptors to trigger growth hormone release while preserving natural production. Achieves superior oral bioavailability exceeding 60% with a 24-hour half-life, making it unique among GH secretagogues for its convenient once-daily oral dosing.
Moleküler Veri
Araştırma Endikasyonları
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Doz Protokolleri
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| Hedef | Doz | Sıklık | Yol |
|---|---|---|---|
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Etkileşimler
CJC-1295
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Ipamorelin
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GHRP-2
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HGH
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LGD-4033
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Yan Etkiler & Güvenlik
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Kaynaklar
- Effects of a 7-day treatment with a novel, orally active, growth hormone (GH) secretagogue, MK-677, on 24-hour GH profiles, insulin-like growth factor I, and adrenocortical function in normal young men — Copinschi, G., et al.
- Stimulation of the growth hormone (GH)-insulin-like growth factor I axis by daily oral administration of a GH secretagogue (MK-677) in healthy elderly subjects — Chapman, I.M., et al.
- Prolonged oral treatment with MK-677, a novel growth hormone secretagogue, improves sleep quality in man — Copinschi, G., et al.
- MK-677, an orally active growth hormone secretagogue, reverses diet-induced catabolism — Murphy, M.G., et al.
- Two-month treatment of obese subjects with the oral growth hormone (GH) secretagogue MK-677 increases GH secretion, fat-free mass, and energy expenditure — Chapman, I.M., et al.
- Oral administration of the growth hormone secretagogue MK-677 increases markers of bone turnover in healthy and functionally impaired elderly adults — Murphy, M.G., et al.
- Effects of an oral ghrelin mimetic on body composition and clinical outcomes in healthy older adults: a randomized trial — Nass, R., et al.