Testosterone
Anabolic-Androgenic Steroid | Primary Male Sex Hormone
Testosterone is the primary endogenous androgenic-anabolic steroid hormone produced mainly by the Leydig cells of the testes in males and in smaller quantities by the ovaries and adrenal glands in females. It is essential for the development and maintenance of male reproductive tissues, secondary sexual characteristics, muscle mass, bone density, red blood cell production, and overall well-being. Exogenous testosterone has been FDA-approved for the treatment of male hypogonadism since the 1950s and remains the gold standard for testosterone replacement therapy (TRT). It is available in multiple pharmaceutical formulations including intramuscular injectables, transdermal gels, transdermal patches, subcutaneous pellets, and oral capsules. In supraphysiological doses, testosterone is also widely used for performance enhancement, though such use falls outside approved medical indications.
Moleküler Gösterim
M.W.: 288.42 Da (base)
PubChem 2D yapı diyagramı
Referans Flakon
Referans illüstrasyonu — ürün listesi değildir
Etki Mekanizması
Testosterone exerts its effects primarily through binding to the intracellular androgen receptor (AR), forming a hormone-receptor complex that translocates to the nucleus and modulates gene transcription. This drives protein synthesis in skeletal muscle (anabolic effect), stimulates erythropoietin production in the kidneys to increase red blood cell mass, promotes osteoblast activity and bone mineral density, and regulates libido and cognitive function. Testosterone is also converted to dihydrotestosterone (DHT) by the enzyme 5-alpha reductase in peripheral tissues (skin, prostate, hair follicles), where DHT mediates androgenic effects with greater potency. Additionally, testosterone is aromatized to estradiol by the enzyme aromatase in adipose tissue, which is important for bone health, lipid metabolism, and cardiovascular function but can cause estrogenic side effects at supraphysiological doses.
Testosterone is the primary endogenous androgenic-anabolic steroid hormone produced mainly by the Leydig cells of the testes in males and in smaller quantities by the ovaries and adrenal glands in females. It is essential for the development and maintenance of male reproductive tissues, secondary sexual characteristics, muscle mass, bone density, red blood cell production, and overall well-being. Exogenous testosterone has been FDA-approved for the treatment of male hypogonadism since the 1950s and remains the gold standard for testosterone replacement therapy (TRT). It is available in multiple pharmaceutical formulations including intramuscular injectables, transdermal gels, transdermal patches, subcutaneous pellets, and oral capsules. In supraphysiological doses, testosterone is also widely used for performance enhancement, though such use falls outside approved medical indications.
Moleküler Veri
Araştırma Endikasyonları
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Doz Protokolleri
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| Hedef | Doz | Sıklık | Yol |
|---|---|---|---|
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| MYMEMORY WARNING: YOU USED ALL AVAILABLE FREE TRANSLATIONS FOR TODAY. NEXT AVAILABLE IN 10 HOURS 21 MINUTES 31 SECONDS VISIT HTTPS://MYMEMORY.TRANSLATED.NET/DOC/USAGELIMITS.PHP TO TRANSLATE MORE | 50-200 mg daily | MYMEMORY WARNING: YOU USED ALL AVAILABLE FREE TRANSLATIONS FOR TODAY. NEXT AVAILABLE IN 11 HOURS 04 MINUTES 04 SECONDS VISIT HTTPS://MYMEMORY.TRANSLATED.NET/DOC/USAGELIMITS.PHP TO TRANSLATE MORE | MYMEMORY WARNING: YOU USED ALL AVAILABLE FREE TRANSLATIONS FOR TODAY. NEXT AVAILABLE IN 10 HOURS 21 MINUTES 31 SECONDS VISIT HTTPS://MYMEMORY.TRANSLATED.NET/DOC/USAGELIMITS.PHP TO TRANSLATE MORE |
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Etkileşimler
HCG
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Anastrozole
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Finasteride
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BPC-157
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Growth Hormone
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CJC-1295/Ipamorelin
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Nandrolone
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Enclomiphene
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Clomiphene
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Ne Beklenmeli
Yan Etkiler & Güvenlik
Yaygın Yan Etkiler
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Durdurma Belirtileri
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Kontrendikasyonlar
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Sık Sorulan Sorular
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Kaynaklar
- Testosterone Therapy in Men With Hypogonadism: An Endocrine Society Clinical Practice Guideline — Bhasin, S., Brito, J.P., Cunningham, G.R., et al.
- Effects of Testosterone Treatment in Older Men — Snyder, P.J., Bhasin, S., Cunningham, G.R., et al.
- Testosterone Treatment and Cardiovascular Events in Men with Low Testosterone: The TRAVERSE Randomized Clinical Trial — Lincoff, A.M., Bhasin, S., Flevaris, P., et al.
- Testosterone dose-response relationships in healthy young men — Bhasin, S., Woodhouse, L., Casaburi, R., et al.
- Testosterone Replacement Therapy and Cardiovascular Risk: A Review — Corona, G., Torres, L.O., Maggi, M.