Retatrutide
Triple GLP-1/GIP/Glucagon Agonist | Weight Loss & Diabetes
Novel triple hormone receptor agonist targeting GLP-1, GIP, and glucagon receptors. Phase II trials demonstrated 24.2% weight loss at 48 weeks—the highest recorded for obesity medications.
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M.W.: 4,731.33 Da
PubChem 2D yapı diyagramı
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Referans illüstrasyonu — ürün listesi değildir
Etki Mekanizması
Activates GLP-1 for appetite suppression, GIP for insulin sensitivity, and glucagon for increased energy expenditure and hepatic fat oxidation.
Novel triple hormone receptor agonist targeting GLP-1, GIP, and glucagon receptors. Phase II trials demonstrated 24.2% weight loss at 48 weeks—the highest recorded for obesity medications.
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Kaynaklar
- Triple-Hormone-Receptor Agonist Retatrutide for Obesity — A Phase 2 Trial — Jastreboff, A.M., et al.
- Retatrutide, a GIP, GLP-1 and glucagon receptor agonist, for people with type 2 diabetes: a phase 2 trial — Rosenstock, J., et al.
- Triple hormone receptor agonist retatrutide for metabolic dysfunction-associated steatotic liver disease: a randomized phase 2a trial — Sanyal, A.J., et al.
- Structural insights into the triple agonism at GLP-1R, GIPR and GCGR manifested by retatrutide — Li, W., et al.
- TRIUMPH registrational clinical trials: Rationale and design — Aronne, L.J., et al.
- Effects of retatrutide on body composition in people with type 2 diabetes: a phase 2 substudy — Rosenstock, J., et al.